[1,2,4]Triazolo[3,4-b]benzothiazole Scaffold as Versatile Nicotinamide Mimic Allowing Nanomolar Inhibition of Different PARP Enzymes

Murthy, Sudarshan.; Nizi, Maria Giulia; Maksimainen, Mirko M.; Massari, Serena.; Alaviuhkola, Juho.; Lippok, Barbara E.; Vagaggini, Chiara.; Sowa, Sven T.; Galera-Prat, Albert.; Ashok, Yashwanth.; Venkannagari, Harikanth.; Prunskaite-Hyyrylaeinen, Renata.; Dreassi, Elena.; Luscher, Bernhard.; Korn, Patricia.; Tabarrini, Oriana. (Corresponding author); Lehtio, Lari. (Corresponding author)

Washington, DC : ACS (2023)
Journal Article

In: Journal of medicinal chemistry
Volume: 66
Issue: 2
Page(s)/Article-Nr.: 1301-1320